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Data / Drug companies / Opioid Antagonist

Opioid Antagonist drugs: 22 drugs from 95 companies in the FDA NDC directory

Opioid Antagonist is an FDA established pharmacologic class. The FDA National Drug Code Directory lists 267 products in this class from 95 companies, covering 22 drugs by generic name. The main marketing category is generic drugs (ANDA), and the newest product started marketing on October 28, 2026.

SpecStream is the live web data engine for teams and agents. It reads the National Drug Code Directory that FDA publishes, and this page is that reading. Ask for the companies that make a drug, a class or a dosage form, with their headquarters, website and size added from the web, and new listings and discontinued products arrive in your sheet, CRM, Slack or agent as FDA posts them.

  • 95Companies
  • 267Products
  • 22Drugs by generic name

Drugs in the Opioid Antagonist class

Ranked by number of companies that list the drug.

DrugProducts hereCompanies listing it
Naloxone hydrochloride8040
Naltrexone hydrochloride4524
Buprenorphine and naloxone6522
Alvimopan44
Buprenorphine hydrochloride and naloxone hydrochloride143
Nalxone hydrochloride43
Naloxone hcl33
Naloxone hydrochloride nasal33
Nalmefene hydrochloride32
Naloxegol oxalate32
Pentazocine hydrochloride and naloxone hydrochloride22
Buprenorphine hydrochloride, naloxone hydrochloride41
Olanzapine and samidorphan l-malate41
Methylnaltrexone bromide31
Nalmefene hydrochloride injection21
Naldemedine11
Naloxone11
Naloxone hci11
Naltrexone hydrochloride and bupropion hydrochloride11
Narcan naloxone hci11
Narcan naloxone hcl11
Pentazocine and naloxone11

Companies with the most products in this class

CompanyProductsMain dosage formsMain marketing categoryNewest product started
Bryant Ranch Prepack22tablet, film coated; tabletGeneric drugs (ANDA)August 15, 2025
HF Acquisition Co LLC, DBA HealthFirst15injection, solution; injectionGeneric drugs (ANDA)August 28, 2023
Medical Purchasing Solutions, LLC9injection, solution; injectionGeneric drugs (ANDA)January 29, 2021
A-S Medication Solutions8spray; injection, solutionGeneric drugs (ANDA)July 30, 2023
Redpharm Drug8film; tabletGeneric drugs (ANDA)August 29, 2023
Bryant Ranch Prepack7tablet, film coated; tabletGeneric drugs (ANDA)August 15, 2025
Remedyrepack Inc.7tablet; tablet, film coatedGeneric drugs (ANDA)October 28, 2026
Camber Pharmaceuticals, Inc.6film, soluble; tabletGeneric drugs (ANDA)May 1, 2026
Edenbridge Pharmaceuticals LLC.6tablet, orally disintegratingNew drug applications (NDA)June 12, 2026
Orexo US, Inc.6tablet, orally disintegratingNew drug applications (NDA)December 11, 2014
Bryant Ranch Prepack5tablet; tablet, film coatedGeneric drugs (ANDA)April 13, 2020
Clinical Solutions Wholesale, LLC5tabletGeneric drugs (ANDA)September 1, 2020
Dr. Reddy's Laboratories Inc.5film, soluble; injectionGeneric drugs (ANDA)March 18, 2020
Indivior Inc.5film, soluble; sprayNew drug applications (NDA)October 2, 2023
Alkermes, Inc.4tablet, film coatedNew drug applications (NDA)September 20, 2021
Alvogen Inc.4filmGeneric drugs (ANDA)February 11, 2019
Aveva Drug Delivery Systems Inc.4filmGeneric drugs (ANDA)March 7, 2025
Golden State Medical Supply, Inc.4tablet; capsuleGeneric drugs (ANDA)August 31, 2023
Hikma Pharmaceuticals USA Inc.4injectionGeneric drugs (ANDA)July 25, 2025
Ingenus Pharmaceuticals, LLC4filmGeneric drugs (ANDA)August 29, 2023
International Medication Systems, Limited4injection; sprayGeneric drugs (ANDA)May 7, 2024
Mylan Pharmaceuticals Inc.4filmGeneric drugs (ANDA)April 17, 2020
Accord Healthcare Inc.3tablet; tablet, film coatedGeneric drugs (ANDA)September 1, 2020
Actavis Pharma, Inc.3capsule; tabletGeneric drugs (ANDA)January 17, 2025
Eugia US LLC3injection, solutionGeneric drugs (ANDA)January 14, 2021
Henry Schein, Inc.3injection, solution; injectionGeneric drugs (ANDA)October 28, 2025
Hikma Pharmaceuticals USA Inc.3tablet; capsuleGeneric drugs (ANDA)February 6, 2024
Hospira, Inc.3injection, solutionGeneric drugs (ANDA)September 23, 2005
Major Pharmaceuticals3tablet; tablet, film coatedGeneric drugs (ANDA)June 27, 2014
Mylan Institutional LLC3injection, solutionGeneric drugs (ANDA)December 2, 2022
Salix Pharmaceuticals, Inc.3injection, solution; tabletNew drug applications (NDA)August 1, 2008
SpecGx LLC3tablet; tablet, film coatedGeneric drugs (ANDA)December 13, 2017
Unit Dose Solutions, Inc.3tabletGeneric drugs (ANDA)April 13, 2026
Actavis Pharma, Inc.2tabletGeneric drugs (ANDA)March 4, 2013
American Health Packaging2tabletGeneric drugs (ANDA)March 14, 2022
Amneal Pharmaceuticals LLC2tabletGeneric drugs (ANDA)February 22, 2013
Aphena Pharma Solutions - Tennessee, LLC2tablet, film coatedGeneric drugs (ANDA)March 22, 2002
Aphena Pharma Solutions - Tennessee, LLC2tablet, film coatedGeneric drugs (ANDA)August 15, 2025
Ascend Laboratories, LLC2tabletGeneric drugs (ANDA)July 3, 2026
Asclemed USA, Inc.2spray, metered; tabletGeneric drugs (ANDA)September 23, 2024
AvKARE2tablet, film coated; sprayGeneric drugs (ANDA)May 1, 2024
AvPAK2tabletGeneric drugs (ANDA)December 8, 2016
Averitas Pharma, Inc.2tablet, film coatedNew drug applications (NDA)March 28, 2023
Baxter Healthcare Corporation2injection, solutionGeneric drugs (ANDA)November 7, 2022
Chengdu Shuode Pharmaceutical Co., Ltd2solutionGeneric drugs (ANDA)November 15, 2023
Coupler LLC2tablet, film coatedGeneric drugs (ANDA)June 15, 2026
Emergent Devices Inc.2sprayNew drug applications (NDA)August 28, 2023
Fresenius Kabi USA, LLC2injection, solutionGeneric drugs (ANDA)April 2, 2024
Knoa Pharma LLC2injection, solutionNew drug applications (NDA)August 7, 2025
Lannett Company, Inc.2tabletGeneric drugs (ANDA)September 19, 2016
Lifestar Pharma LLC2injection, solutionGeneric drugs (ANDA)February 19, 2026
Pai Holdings, LLC DBA Pai Pharma2tabletGeneric drugs (ANDA)September 5, 2023
Precision Dose, Inc.2tablet, film coatedGeneric drugs (ANDA)February 15, 2024
ProPharma Distribution2injection, solutionGeneric drugs (ANDA)August 8, 2017
Proficient Rx LP2sprayNew drug applications (NDA)June 21, 2022
Rhodes Pharmaceuticals LLC2tabletGeneric drugs (ANDA)April 13, 2020
Somerset Therapeutics, LLC2injection, solutionGeneric drugs (ANDA)August 8, 2017
Sportpharm LLC2spray, metered; sprayGeneric drugs (ANDA)September 23, 2024
Sun Pharmaceutical Industries, Inc.2tabletGeneric drugs (ANDA)July 18, 2017
Advanced Rx of Tennessee, LLC1sprayGeneric drugs (ANDA)June 27, 2024
American Health Packaging1tablet, film coatedGeneric drugs (ANDA)June 3, 2013
Amerisource Bergen1sprayGeneric drugs (ANDA)March 12, 2025
Amneal Pharmaceuticals NY LLC1sprayGeneric drugs (ANDA)April 24, 2024
Amneal Pharmaceuticals NY LLC1sprayGeneric drugs (ANDA)April 24, 2024
Baxter Healthcare Corporation1injection, solutionGeneric drugs (ANDA)June 3, 2025
BioDelivery Sciences International Inc1tabletNew drug applications (NDA)June 14, 2019
BluePoint Laboratories1sprayGeneric drugs (ANDA)May 1, 2025
Bpi Labs LLC1injection, solutionGeneric drugs (ANDA)November 15, 2023
CVS Woonsocket Prescription Center, Incorporated1sprayGeneric drugs (ANDA)April 24, 2024
Chartwell RX, LLC1tablet, film coatedGeneric drugs (ANDA)July 21, 2017
Civica, Inc.1injectionGeneric drugs (ANDA)November 11, 2019
Elite Laboratories, Inc.1tablet, film coatedGeneric drugs (ANDA)August 15, 2025
Harm Reduction Therapeutics, Inc.1sprayNew drug applications (NDA)January 2, 2024
Heritage Pharmaceuticals Inc. D/B/A Avet Pharmaceuticals Inc.1tablet, film coatedGeneric drugs (ANDA)October 6, 2023
Hikma Specialty USA Inc.1sprayNew drug applications (NDA)August 3, 2021
Kaleo, Inc1injection, solutionNew drug applications (NDA)February 28, 2022
Lupin Pharmaceuticals,Inc.1tabletGeneric drugs (ANDA)May 11, 2011
NCS HealthCare of Ky, LLC DBA Vangard Labs1tablet, film coatedGeneric drugs (ANDA)February 29, 2012
Nalpropion Pharmaceuticals LLC1tablet, extended releaseNew drug applications (NDA)October 22, 2014
NorthStar RxLLC1injection, solutionGeneric drugs (ANDA)July 1, 2024
NuCare Pharmaceuticals,Inc.1tablet, film coatedGeneric drugs (ANDA)February 15, 2024
Padagis Israel Pharmaceuticals Ltd1sprayGeneric drugs (ANDA)July 30, 2023
Par Health USA, LLC1injectionGeneric drugs (ANDA)November 5, 2024
Par Health USA, LLC1capsuleGeneric drugs (ANDA)May 3, 2023
Proficient Rx LP1tablet, film coatedGeneric drugs (ANDA)February 29, 2012
RedHill Biopharma Ltd1tablet, film coatedNew drug applications (NDA)October 1, 2020
Scienture LLC1sprayNew drug applications (NDA)January 29, 2026
Sina Health Inc1injection, solutionGeneric drugs (ANDA)August 8, 2017
Strategic Sourcing Services LLC1sprayGeneric drugs (ANDA)April 1, 2025
Sun Pharmaceutical Industries, Inc.1tabletGeneric drugs (ANDA)July 31, 2018
Sun Pharmaceutical Industries, Inc.1tablet, film coatedGeneric drugs (ANDA)February 29, 2012
Tagi Pharma, Inc.1tablet, film coatedGeneric drugs (ANDA)September 23, 2013
Teva Pharmaceuticals, Inc.1spray, meteredGeneric drugs (ANDA)September 23, 2024
Walgreen Company1sprayGeneric drugs (ANDA)April 24, 2024
Zmi Pharma Inc.1injection, solutionNew drug applications (NDA)January 15, 2022

Dosage forms

Dosage formProductsShare
Tablet6424%
Tablet, film coated5219.5%
Injection, solution4717.6%
Spray2810.5%
Film217.9%
Injection197.1%
Film, soluble124.5%
Tablet, orally disintegrating124.5%
Capsule41.5%
Spray, metered41.5%
Solution20.7%
Inhalant10.4%

Updated November 6, 2026. Read from US Food and Drug Administration, National Drug Code Directory (openFDA). CC0 1.0 public domain dedication (openFDA). Counts are products in the FDA National Drug Code Directory on November 6, 2026: 138,262 products in commercial distribution, meaning without a marketing end date in the past. A company is a labeler code; one company can hold several codes, and the directory carries no address. Inclusion in the directory is not FDA approval, and the marketing category says under which kind of application or rule a product is sold. This page uses openFDA data and is not endorsed or certified by FDA. Free to reuse with credit to SpecStream under CC BY 4.0. Spot a wrong value? Write to [email protected] with the link to this page.